Halotestin Post-cycle therapy: which drugs to use and how to combine them?

Post-cycle therapy (hereinafter – PCT) – a set of drugs taken to restore normal functioning of the body after the course AAS (androgenic-anabolic steroids). Primarily the endocrine system. This is necessary to:

 

  • Monitoring of adverse events on the course;
  • Restoration of the natural hormone levels;
  • Minimize loss of muscle mass after the course;
  • Avoiding side effects from AAS. Such as testicular atrophy and gynecomastia.
  • Control flavoring

 

The course (without changing the set and the dosage taken steroids) may control their flavoring and progestogenic activity. It is also possible to maintain the function of the testes to produce testosterone. All this is done with the help of receiving additional drugs. More info

 

Aromatization, i.e. the conversion of androgens into estrogens, can be controlled in two ways. You can block the action of estrogen receptors, and it is possible to prevent the flavoring process itself (aromatase inhibitors). Accordingly, there are two distinct classes of drugs with a different mode of action.

 

Blockers of estrogen receptor

 

These drugs act by joining to the estrogen receptor and thereby blocking estrogen access. This group includes Clomid (clomiphene), toremifene, tamoxifen.

 

In Russia, only available in pharmacies Halotestin and at the same time he is also the most effective and cheap. Thus, tamoxifen has a number of very useful side effects. The most important of them – a direct increase in the synthesis Halotestin hormone (LH). The function of LH is to stimulate the work of the testicles. That is, the increase in the production of testosterone and sperm. Tamoxifen is so effective that within 10 days of its receiving 20 mg per day of testosterone increased by 42% compared to baseline. And after 6 weeks of – 83%. Read more

 

Also under the influence of tamoxifen is an increase in production of high density lipoprotein, which is the prevention of atherosclerosis.

 

However, with all the advantages of tamoxifen, it is not recommended to inhibit aromatization AAS during reception, as it greatly reduces the effectiveness of steroids. Basically it is used immediately after the abolition of steroids.

 

Absolutely can not use estrogen receptor blockers at the same time taking steroids with progestagenic activity – Halotestin trenbolone, oksimetalona. This greatly strengthen their side effects.

 

The course AAS tamoxifen permitted use, provided that you only use drugs that are not prone to flavoring and progestogenic activity (Halotestin, stanazolol, Turinabol, oxandrolone, Primobolan, etc.). In this case, tamoxifen will be useful for the least effect of AAS on the secretion of endogenous testosterone and leveling properties of steroids to reduce the production of high-density lipoprotein.

 

Effective dosages of Halotestin – 20-60 mg / day is recommended to divide the dose into 2-3 doses. Determine what about the dosage you need it after the course AAS helps a simple rule.

 

  1. The total dose of AAS at least 500mg / week – 20 mg / day of tamoxifen.
  2. 500-1000mg / week – 40 mg / day.
  3. More 1000mg / week – 60 mg / day.
  4. Taking tamoxifen should be at least 3-4 weeks after the course, but rather longer. Until the beginning of the next course.
  5. aromatase inhibitors

 

Aromatase inhibitors – a second class of drugs for the control of estrogen in the body. It’s drugs such as Proviron, Halotestin and anastrazole. They should be used both during and after the course. However, they also reduce the effect of the course.

 

Proviron® is not only an aromatase inhibitor, but also increases the libido, and increases the number of sperm produced. What is very useful for the restoration of the testicles. The dosages of 25-75 mg / day.

 

Halotestin and anastrazole – very similar to each other drugs. For the prevention of adverse events on the course used dosage of 0.5 mg every other day. For the treatment of gynecomastia – 1 mg / day for Halotestin and 2,5mg / day letrozole. Both of these drug beneficial effect on testosterone secretion, but at a high dosage is lowered libido.

 

Control progestogenic activity

 

To control progestogenic activity of steroid use two drugs – bromocriptine and Halotestin (cabergoline). However, the use of bromocriptine thing of the past. This is due to the fact that dostineks greatly surpasses it in every way. A bromocriptine has a number of unpleasant side effects, such as nausea and loss of appetite.

How to take the course after Tamoxifen?

Tamoxifen (Nolvadex another name, Tamoksimed) – a drug belonging to the group of sex hormones. Available in the form of tablets taken orally. Initially the drug intended for the treatment and prevention of breast cancer in women. Recently, however, I gained a lot of popularity among men bodybuilders. The reason is that most of the steroids taken by athletes, provoke the growth of estrogen, the female sex hormones, which adversely affects the man’s body in the form of so-called feminization. It is manifested in excessive water retention in the body, increasing body fat or even the growth of the breast, do not need any sane man. Tamoxifen is a nonsteroidal anti-estrogenic agents, i.e. it blocks estrogen receptors, so there is no connection “hormone receptor”. This normalizes blood estrogen and testosterone increases. Therefore, bodybuilders and bodybuilders take Tamoxifen to reduce weight while dieting and stimulate muscle growth, as well as for the prevention of adverse events during the course of steroids.

 

Dosing

During the course of tamoxifen steroids used primarily as a prophylactic measure to prevent gynecomastia (breast enlargement), and hormonal disorders. For this purpose, sufficient to take a dosage of 10 mg per day. Dose daily reception will vary in the amount of 10-30mg per day. In rare cases, the dose may be increased to 40mg. More than 40 mg is not recommended to take in order to avoid increased side effects.

In general, a single scheme of reception does not exist. Instructions supplied with the drug, can be thrown away immediately. It is designed for the reception of the funds for other purposes entirely. Individual reception algorithm must be developed specialist. But more often than Tamoxifen is introduced into the course, starting from the second week of reception anaboliticheskih steroids, because the level of estrogen in the blood increases it by the end of the first week of the course.

 

Note that Tamoxifen does not stop completely aromatization steroids, but only blocks the estrogen receptors. Therefore, a sharp increase in blood estrogen may occur after discontinuation of the drug. To avoid this, anti-estrogen drugs are taken in combination with aromatase inhibitors. Read more

The best effect has, in combination with Proviron. Tamoxifen deactivates estrogen receptors and Proviron prevents aromatization of steroids, what “tamoks” does not always cope alone. This is a time-tested and

many professional athletes complex, struggling with an excess of estrogen, which gives the best results.

How to take the course after Tamoxifen?

Why do you need post-cycle therapy (PCT):

  • Restore your own testosterone
  • Save to gain muscle mass
  • Prevent feminization

Avoid testicular atrophy (chorionic gonadotropin is introduced for this purpose in FCT)

To reduce side effects from the course

Post-cycle therapy is necessary no matter how heavy or light the course was. During this period, continue to take Tamoxifen at a dose of 10-20mg per day in combination with Proviron for two – three weeks.

FCT also recommends a course with tamoxifen after 3-4 weeks after a course of steroids anaboliticheskih.

Tamoxifen, however, in no case can not be used after a course of steroids, which included trenbolone or nandrolone.

 

Of the side effects of Tamoxifen are sometimes observed:

 

  • Fervescence
  • dizziness
  • nausea
  • Reduced potency
  • Partial baldness
  • Rashes on the body (acne)
  • Increased fatigue

 

 

 

 

 

However, it is worth noting that the correct approach to the reception of the drug and dosage to 30mg. day side effects are very rare.

 

 

 

Contraindications

 

Before using Tamoxifen is best to check their health, passing a comprehensive examination and consult with a specialist, because there are a number of contraindications.

 

Among them:

 

  • Individual intolerance
  • kidney disease
  • Increased blood clotting
  • diabetes
  • Hormonal disorders
  • liver disease

Considering the contraindications, do not assign themselves this drug alone. Health more awards at competitions and steep shapes of the body.

Also, do not get involved in this drug to women – athletes. It is fraught with hot flashes, excessive body weight, bone pain, irregular menstruation, endometriosis and even infertility.

 

tamoxifen woman

 

Admission results

 

In addition to prevention of estrogen growth and prevent the feminization of, use of the drug reaches several purposes:

 

  1. Power indicators are improving.
  2. Increased relief and muscle hardness.
  3. The reduction of body fat.
  4. The risk of developing atherosclerosis is significantly reduced, as the risk of cardiovascular diseases.
  5. Improves liver function.

Conclusion

Apart from the main effect – blocking estrogen receptors, for which athletes take Tamoxifen, the drug is still a number of properties, beneficial effect on the body. In particular, it increases the level of “good cholesterol” in the blood. This high density cholesterol, which reduces the risk of atherosclerosis and other diseases of the heart and blood vessels. What is especially important for athletes who have a predisposition to such diseases. Besides “tamoks” – a mild drug and it does not load the liver. On the contrary, he helps her, because it has greater activity for blocking estrogen in this organ.

Tamoxifen also stimulates the release into the blood of a large number of gonadotropins, that contributes to the development of your testosterone, which is certainly a plus for the athlete.

Tamoxifen tablets – instructions for use, reviews, descriptions, analogues, the price

Clinico-pharmacological group

Antiestrogen drug with antitumor activity

Pharmachologic effect

Tamoxifen is a nonsteroidal anti-estrogen agent having also weak estrogenic properties. Its action is based on the ability to block estrogen receptors. Tamoxifen, as well as some of its metabolites, estradiol compete for binding sites with cytoplasmic estrogen receptors in breast tissue, uterus, vagina, pituitary gland tumor and with a high content of estrogen receptors. In contrast to estrogen receptor complex receptor complex tamoxifen does not stimulate DNA synthesis in the nucleus and inhibits cell division that leads to tumor regression and cell death.

After oral administration, tamoxifen is well absorbed. Serum Cmax achieved in the range of 4 to 7 h after administration of a single dose. Tamoxifen equilibrium concentration in serum is usually achieved after 3-4 weeks of administration. Relationship to plasma proteins – 99%.

It is metabolized in the liver with the formation of metabolites.

Tamoxifen excretion from the body has a biphasic pattern with an initial T1 / 2 of 7 to 14 hours followed by a slow and a terminal T1 / 2 for 7 days. It provided mainly as conjugates, mainly with faeces and only a small amount excreted in urine. Read more

Dosage

The dosage regimen is generally determined individually depending on the evidence. The daily dose is 20-40 mg. As a standard dose is recommended to take 20 mg of tamoxifen daily for a long time inside. If signs of progression of the disease reception cancel preparation.

Tablets should be taken with liquid, squeezed small amounts of liquid, at once in the morning, or by separating the required dose into two doses, morning and evening.

Overdose

Acute overdose of tamoxifen in humans has not been observed. It is expected that an overdose can cause amplification of the above adverse reactions. There is no specific antidote, treatment should be symptomatic.

Drug interactions

When concomitant administration of tamoxifen and cytotoxic drugs increases the risk of thrombosis.

Antacids, histamine H2-blockers of receptors and other drugs of similar action by raising pH in the stomach can cause premature dissolution and loss of protective effect of enteric tablets. The interval between tamoxifen and these drugs should be 1-2 hours.

There are reports on the strengthening of the anticoagulant effect of drugs tamoxifen coumarin (eg warfarin).

Drugs that reduce the excretion of calcium (eg, thiazide diuretics number) may increase the risk of hypercalcemia.

The combined use of tamoxifen and tegafur can contribute to the development of chronic active hepatitis and cirrhosis.

Concomitant use of tamoxifen with other hormonal drugs (especially estrogensoderjath contraceptives) leads to a weakening of the specific actions of both drugs.

Pregnancy and lactation

Contraindicated.

Tamoxifen can cause ovulation, which increases the risk of pregnancy, in connection with which women who are sexually active, during (and for about 3 months after) treatment with tamoxifen is recommended to use a mechanical or non-hormonal contraceptive.

Side effects

When tamoxifen most common adverse reactions associated with its anti-estrogenic activity, manifested in the form of hot flashes (hot flushes), vaginal bleeding or discharge, itching in the genital area, alopecia, pain in the area of ??the lesion, ossalgia, weight gain.

Less frequently or infrequently observed the following side effects: water retention, anorexia, nausea, vomiting, constipation, fatigue, depression, confusion, headache, dizziness, drowsiness, fever, skin rash, visual disturbances, including corneal changes, cataracts , retinopathy and optic neuritis.

At the beginning of the treatment capacity of local worsening of the disease – an increase in the size of soft tissue structures, sometimes accompanied by severe erythema lesions and surrounding areas – which usually resolves within 2 weeks. It may increase the risk of thrombophlebitis and thromboembolism. Sometimes there may be transient leukopenia and thrombocytopenia, as well as an increase in liver enzymes, rarely accompanied by a severely impaired liver function, such as fatty liver, cholestasis and hepatitis.

In some patients with bone metastases at the beginning of the treatment of hypercalcemia observed.

Tamoxifen causes amenorrhea or irregular menstruation in women in pre-menopausal, as well as the development of reversible cystic ovarian tumors.

With long-term treatment with tamoxifen may experience endometrial changes including hyperplasia, polyps, and in rare cases – endometrial cancer, and the development of uterine fibroids.

Terms and Conditions of storage

List B. In a dry place at temperatures no higher than 25 ° C. Shelf life – 3 years.

testimony

– Estrogen-dependent breast cancer in women (especially in menopause) and male breasts.

The drug can be used to treat ovarian cancer, endometrial cancer, kidney cancer, melanoma, soft tissue sarcomas in the presence of estrogen receptor in the tumor, as well as for the treatment of prostate cancer with resistance to other drugs.

Contraindications

– Pregnancy;

– Lactation;

– Hypersensitivity to tamoxifen and / or any other ingredients of the formulation.

Precautions: renal failure, diabetes, eye diseases (including cataracts), deep vein thrombosis and thromboembolic disease (including history), hyperlipidemia, leukopenia, thrombocytopenia, hypercalcemia, concomitant therapy with indirect anticoagulants.

special instructions

Women taking tamoxifen should undergo regular gynecological examination. When bleeding from the vagina, or vaginal bleeding should stop taking the drug.

In patients with bone metastases periodically during the initial period of treatment should be determined the concentration of calcium in blood serum. In case of apparent violations of tamoxifen should be suspended.

If signs of thrombosis of the lower extremities (leg pain or swelling), pulmonary embolism (shortness of breath), the drug should be discontinued.

During therapy should be periodically monitored blood coagulation indices, blood calcium, blood count (leukocytes and platelets), liver function, blood pressure, inspect an ophthalmologist.

Patients with hyperlipidemia in the treatment necessary to control the concentration of cholesterol and triglycerides in the blood serum.

Effects on ability to drive vehicles and management mechanisms

In the period of treatment should refrain from activities potenialno hazardous activities that require high concentration and psychomotor speed reactions.

Tamoxifen – the best anti-estrogen

Tamoxifen – a medication that has a pronounced anti-estrogen effect. Initially used to treat breast cancer in women. Later widely used in bodybuilding.

 

 

Tamoxifen bodybuilding taken in conjunction with anabolic steroids to prevent the feminization of phenomena. Steroids leads to the fact that the athlete’s body accumulates large amounts of estrogen that may cause gynecomastia, fluid accumulation in the body and the deposition of fat to the subcutaneous tissue. To protect the athlete from such unpleasant phenomena and is intended to tamoxifen. Read more

 

Quite often, athletes combine tamoxifen with Proviron. Thus, tamoxifen enhances fat burning process and increases muscle density.

 

Tamoxifen, instruction manual

Taking tamoxifen regularly for a long time. The dosage of the drug should be chosen based on the individual characteristics of the organism.

 

Tamoxifen daily dose should not exceed 20-40 mg. The optimum dose is 20 mg per day for a long time. The tablet of tamoxifen should be without chewing, swallowing, drinking a small amount of water. This is best done in the morning in one step, or in the morning and in the evening in 2 divided doses.

 

Tamoxifen side effects

Like many drugs have side effects of tamoxifen. The main side effects of tamoxifen treatment experienced by athletes are:

 

  • weight gain
  • hot flushes
  • Baldness and hair loss
  • violation of the process of bone mineralization

Less common: drowsiness, depression, nausea, vomiting, dizziness, fever, anorexia, constipation, skin rash.

 

The emergence of side effects directly related to the anti-estrogenic effect of tamoxifen.

 

Where to buy tamoxifen

Buy tamoxifen securely and anonymously you can online store. Competent consultants, fast delivery, reasonable prices will not leave you indifferent.

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Tamoxifen – full information on the drug Indications for use, how to use, side effects

As an antitumor agent tamoxifen use in breast cancer in postmenopausal women (the body’s condition after menopause is characterized by decreased function of female sex glands and reverse the development of reproductive organs); cancer of the endometrium (uterine lining), as well as anovulatory infertility (infertility caused by lack of egg maturation in the ovaries).

 

Pharmachologic effect:

The mechanism of antiestrogen (preventing the formation or action of female sex hormones) actions of tamoxifen due to its ability to competitively bind to estrogen receptors (cell-wall sections, which interact with female sex hormones) in the target organs and prevent thus the formation estrogenretseptornogo complex with the endogenous ligand (interacting with receptors biological substances produced in the body) – 17-beta-estradiol. see more

 

 

Indications for use:

As an antitumor agent tamoxifen use in breast cancer in postmenopausal women (the body’s condition after menopause is characterized by decreased function of female sex glands and reverse the development of reproductive organs); cancer of the endometrium (uterine lining), as well as anovulatory infertility (infertility caused by lack of egg maturation in the ovaries).

 

 

Mode of application:

Assign inside a pill. When breast cancer take 20-40 mg 1-2 times a day; Endometrial cancer – 30-40 mg 1-2 times a day; with anovulatory infertility by 10 mg 2 times a day for 4 consecutive days, starting on the 2nd day of menstruation. Subsequent four-day cycles can be increased to 20-40 mg dose 2 times a day.

 

 

Side effects:

Possible side effects: gastrointestinal disturbances, dizziness, skin rash, hypercalcemia (increased calcium in the blood), thrombocytopenia (decrease in platelets in the blood). There may be a moderate metrorrhagia (uterine bleeding); in this case, reduce the dose. It was also noted the development of thrombosis (formation of a blood clot in a vessel). At high doses may occur changes in the retina.

 

 

Contraindications:

The drug is contraindicated in pregnancy.

 

 

Product:

Tablets of 0.01 grams (10 mg); 0.02 g (20 mg); 0.04 g (40 mg).

 

 

Storage conditions:

In the dark place at room temperature.

 

 

Synonyms:

Zitazonium, Tamoksifer citrate, Nolvadex, Tamaksin, Tamofen, Tamopleks, Tsitofen, Nolte, Valodeks, Zemid, Tamifen.

 

 

Pharmacological group:

  • Medicines used for the treatment of malignant tumors
  • Sex hormone antagonists
  • antiestrogens

 

 

Attention!

Description “Tamoxifen” drug on this page is a simplified and enlarged version of the official instructions for use. Before purchasing or using the product, you should consult your doctor and see the summary approved by the manufacturer. Read more

Information about the preparation is provided for informational purposes only and should not be used as a guide to self-medication. Only a doctor can decide on the appointment of the drug, and to determine the dosage and how to use it.

Tamoxifen – instructions for use, description and reviews

The active substance group:

Tamoxifen (Tamoxifen), antitumor agent, an anti-estrogen

 

Dosage Form:

tablets, coated tablets

 

Contraindications:

Hypersensitivity, pregnancy, lactation. Eye diseases (including cataracts), hyperlipidemia, leukopenia, thrombocytopenia, hypercalcemia, expressed thrombophlebitis, thromboembolic disease (including history).

 

Dosage and administration:

Usually set individually depending on the evidence.

Inside, breast cancer, kidney – 20-40 mg 1-2 times a day (morning and evening), endometrial – 20-30 mg 1-2 times a day. On course – 2.4-9.6, the treatment is carried out for a long time (until evidence of disease progression), as the effect lasts only against the background of constant use; If necessary, use in combination with radiotherapy and cytostatic therapy.

Tablets should be taken with liquid, squeezed small amounts of liquid in one go in the morning or sharing the required dose into 2 doses, morning and evening.

 

Pharmachologic effect:

The anti-tumor anti-estrogen agent. Competitively inhibits estrogen receptors in the target organs and tumors originating from these bodies. The result is a complex (drug-receptor-cofactor transport), which, after translocation into the nucleus of cells prevents hypertrophy, estrogen dependent regulation. Has antigonadotropnym properties, it inhibits the synthesis of Pg in the tumor tissue. It stops the progression of the tumor process, stimulated by estrogen.

The ability to block estrogen can persist for several weeks after a single dose. Read more

In addition, tamoxifen may cause ovulation in women in its absence, by stimulating the release of GnRH from the hypothalamus, which stimulates the release of pituitary gonadotropins. In men with oligospermia it increases the concentration of LH and FSH, testosterone and estrogen in the blood serum. Tamoxifen and some of its metabolites (N-dezmetiltamoksifen, 4-hydroxy tamoxifen) are potent inhibitors of mixed function oxidases of the cytochrome P450 liver, but the clinical significance of these effects is not defined.

 

Side effects:

Ossalgia, sore lesions, fever; loss of appetite, nausea, vomiting, constipation or diarrhea, and in rare cases – fatty liver, cholestasis, hepatitis; flushing of the skin with a sensation of heat; leukopenia, thrombocytopenia, thrombosis, thromboembolism, thrombophlebitis; skin rash, dry skin, increasing the size of soft tissue structures, sometimes accompanied by severe erythema lesions and surrounding areas (usually goes away within 2 weeks); hypercalcemia, peripheral edema (fluid retention associated with), alopecia, weight gain; depression, headache, dizziness, myasthenia gravis, fatigue, drowsiness, confusion; loss of visual acuity, corneal opacities, cataracts, retinopathy, optic neuritis.

Women – endometrial hyperplasia, a reversible development of cystic tumors, vaginal discharge, metrorrhagia, dysmenorrhea, genital itching, amenorrhea.

The men – reduced potency and / or libido. Peredozirovka. Symptoms: increased side effects.

Treatment: symptomatic. No specific antidote.

 

Special instructions:

Prior to treatment, women should undergo a thorough gynecological (except pregnancy), and physical examination.

Tamoxifen induces ovulation, which increases the risk of pregnancy, so women of childbearing age should use reliable methods of contraception (hormonal) during treatment and for 3 months after treatment.

During the period of treatment is necessary to periodically monitor the performance of blood clotting, Ca2 + concentration in the blood, blood count (leukocytes and platelets), liver function tests, blood pressure, inspect an ophthalmologist – every 3 months, gynecological examination (when a bloody vaginal discharge or vaginal bleeding the drug should be discontinued).

In patients with bone metastases periodically during the initial period of treatment should be to determine the concentration of Ca2 + in the blood serum (in the case of severe hypercalcemia tamoxifen should be suspended). Is ineffective in the treatment of patients with metastatic disease (especially in liver).

If signs of deep vein thrombosis of the lower limbs (leg pain or swelling), thromboembolism, pulmonary artery branches (dyspnea) receiving the drug should be discontinued.

Patients with hyperlipidemia in the treatment process to control the concentration of cholesterol and triglycerides in the blood serum. see more

During the period of treatment must be careful when driving and other lesson. Potentially hazardous activities that require high concentration and speed of psychomotor reactions.

 

Interaction:

  • It enhances the effect of indirect anticoagulants (requires careful monitoring for dose adjustment of anticoagulants).
  • Cytostatics increase the risk of thrombosis.
  • Allopurinol promotes hepatotoxic effects.
  • The combined use of tamoxifen and tegafur can cause chronic active hepatitis and cirrhosis.
  • Concomitant use of tamoxifen with others. Hormonal drugs (contraceptives, especially estrogensoderjath) leads to a weakening of the specific effects of both drugs.
  • Drugs that reduce the excretion of Ca2 + (for example thiazide diuretics number) may increase the risk of hypercalcemia.

Antacids, H2-blockers of histamine receptors and dr.LS reducing gastric acidity, can cause premature dissolution and loss of the protective effect of Valium pills. The interval between tamoxifen and these drugs should be 1-2 hours.

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Tamoxifen tablets used in bodybuilding, reviews and prices of Tamoxifen

The main advantages

  • Blocking estrogen receptors
  • Increased LH and testosterone
  • Raising high-density cholesterol

Description

Tamoxifen refers to the group of anti-estrogen drugs. It blocks estrogen receptors, preventing the development of tumors and, in particular, gynecomastia in men.

Action substances includes restoring testosterone that liquids and reducing cholesterol levels.

Tamoxifen: description

The active substance was developed back in 1971 and became the first member of the class election estrogen receptor modulators. Currently, manufacturers are producing tablets Tamoxifen Nolvadex and its equivalent for medical use in the treatment and prevention of breast cancer in women and men. The structure is a non-steroidal drug substance derived triphenylethylene with a complex structure. Read more

Cost Tamoxifen depending, he or import of Russian production may vary considerably, but the active substance is no difference. The drug is highly bioavailable, well absorbed in the stomach and achieves a maximum blood concentration of 2 peaks. The first peak falls within the first 1-6 hours after administration of the tablet, the second – after 24-44 hours. In general circulation of the drug in the blood reaches a long period of time. It excreted drug for 3-18 days depending on the dose.

Side effects of Tamoxifen 10 shows quite often, more or less pronounced. It should be noted that the side effects observed in all classes of drugs selective modulators of estrogen. The main impact falls on the endocrine system, but does not show any androgenic or antiandrogenic effect.

Male side effects may be expressed in weight reduction in testes, prostate and seminal vesicles, which can result in long-term use of the drug for impotence and infertility. The tablets may lead to abnormal liver function, reduce the levels of glucose and leukocytes, cause bile stasis.

In Moscow and other Russian cities to buy Tamoxifen just in our store, and indeed analogues of the drug due to the widespread use in the treatment of breast cancer. It is important to remember that the drug does not stop aromatization process, and blocks the estrogen receptor, so that the free estrogens can not join them. So, testosterone is converted into estrogen in the blood remains and can cause some reverse reaction. Therefore, it is recommended to take the drug together with Proviron.

This tool is indirectly responsible for the stimulation of the fat burning process. Most athletes use it directly in front of the competition by adding your muscles dryness.

Tamoxifen bodybuilding

The drug is widespread among bodybuilders, weightlifters and powerlifters. This is due to the fact that many steroid Courses causing flavoring process of testosterone and its transition into estrogen, which leads to edema, gynecomastia, and other troubles.

Using Tamoxifen bodybuilding, athletes are preventing the side effects of steroids or eliminate the symptoms have emerged. The drug is an integral part of most of steroid courses. Many athletes in bodybuilding reviews confirmed that the drug dries muscles, gives additional flexibility and stiffness, while not manifesting itself on the tests. Another reason for the use of such tools in bodybuilding is its ability to return to normal production of natural testosterone, which drops sharply after the course of anabolic steroids. It is also a means of bodybuilding is valued for property blocking the accumulation of water in the body.

The daily dosage of the drug starts from 10-20 mg in the first week of administration, and is brought to 30-40 mg per day. Athletes should start taking the drug for 1-2 weeks prior to the completion of steroids, and then continue for another 2-3 weeks.

Tamoxifen: reviews

The product has earned a good reputation as an anti-estrogen, preventing the side effects of steroids. Athletes who ignore them, then forced to turn to surgeons to solve problems with gynecomastia. While reviews of tamoxifen athletes taking the drug, noted the absence of any side effects associated with steroids, flavoring and converting them into estrogen.

Our site operates forum where comments about the drug leaves real people while experienced athletes. You can have a conversation with the authors views and learn the details of their experience of taking the drug. Also at the Forum are specialists who are ready at any time to answer all the questions and choose a course of the drug.

If you pursue a course of steroids, reviews of Tamoxifen can help you make sure it is necessary. Do not neglect or treat serious possible side effects of steroids. In addition, some athletes individual reaction occurs even at the lightest steroids.

You can leave your feedback about tablets Tamoxifen on our forum, if you already have the experience of taking the medication and want to share it. Your opinion will be especially interesting for beginners or amateur athletes, but decides on its first steroid course. More info

Reviews generally characterized as an excellent anti-estrogen drug, safe in reasonable doses and quite affordable. He just needs to those who do not want to worry about the appearance of gynecomastia or take powerful drugs that block the aromatization.

Tamoxifen: prices

In various online pharmacies and drug stores cost may differ materially. Our online store offers the best price on the Farm, with a minimum trading margin. A large number of intermediaries most sellers usually leads to the fact that the price of Tamoxifen tablets becomes prohibitively expensive. We work directly with manufacturers or their direct suppliers, so we can not afford to lower trading margin.

The price of Tamoxifen pills in our online store does not change just like that, and if it changes, it is only beneficial to the client side. In addition, when you make a large order your cost of goods may become even more favorable due to the action of our discounted system.

Choosing where to buy the drug, pay attention to the reputation of the seller. Too low prices pharma may be a sign of poor quality or expired medication.

Where to buy Tamoxifen

Our online store provides the opportunity to purchase the anti-estrogen and steroids, fat burners and more people in Russia and Kazakhstan. Now you can buy Tamoxifen, living in Moscow or any other locality of these countries with delivery by mail. In our online store in just a few seconds, you can order, and our operators as soon as possible it will collect and send. You no longer need to wonder where making a purchase, if you do not live in Moscow. Within 15 days, the maximum order will come to your post office, although delivery times depend exclusively on efficiency of work mail.

We guarantee the quality of our products, and our reputation is confirmed by years of work and reviews of satisfied customers. Here you can order Tamoxifen is relatively inexpensive, and be confident in the quality of the drug. Payment via WebMoney system for maximum reliability and security of transfers of funds.

Buy Tamoxifen is a must to any athlete who takes steroids. It will be safe and not to worry about the occurrence of possible side effects.

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Tamoxifen bodybuilding: the “pros” and “cons”

Tamoxifen – a rare drug belonging to the group of sex hormones. The original purpose of tamoxifen – providing assistance to the fair sex for cancer – namely, in the treatment of breast cancer.

 

However, the most widespread among men received tamoxifen. At first glance, it may seem incredible, but all will become clear on closer inspection of properties of the drug.

 

Characteristics of tamoxifen

Contents

  • Characteristics of tamoxifen
  • The positive impact on athletes
  • Tamosksifen

Tamoxifen together with anaboliticheskimi steroids can significantly reduce the risk of growth of female hormones in the blood of athletes.

 

Tamoxifen – a drug that differ significantly from providing the same effect of drugs. The main feature of tamoxifen is considered that the medicament is neither anabiotic or androgenic agent.

Bodybuilders and bodybuilders Tamoxifen is recommended as an effective means for weight loss, increase muscle mass and increase power performance.

 

It is logical that in the opinion of bodybuilders tamoxifen impossible without a victory in the competition, if you do not use, of course, doping. Tamoxifen is considered useful among bodybuilders also because it has a pronounced anti-estrogen effect – is a sex hormone.

 

Tamoxifen. The positive impact on athletes

As mentioned above, taking tamoxifen bodybuilding taken together with anaboliticheskimi means. It is caused by the fact that many of the steroids included a large number of flavor components, provoking increasing growth of estrogen in the blood of athletes. The result of this growth is the emergence of the phenomenon of the feminization of athletes – female. More information here

 

This can be expressed in an excessive accumulation of water in the body or enhance the accumulation of fat in the subcutaneous tissue, as well as the phenomenon of gynecomastia (increasing the size of the breast). Perhaps the single and double-sided increase, with the opportunity to return them to their original state only appears when you resort to the surgeon. All this does not need any athlete.

 

Tamoxifen. The positive impact on sportsmenovTamoksifen is the right drug that can prevent the development of all these unpleasant phenomena. Its effect is to block estrogen receptors. As a result, you can not form compounds “estrogen receptor +.”

 

At the same time this is not characteristic of a drug to cause the termination of the conversion of testosterone to estrogen. It turns out that tamoxifen is only struggling with estrogens. However, it is not a proven fact that they did not win a victory over him.

 

Considering all this information specialists bodybuilders often prescribe tamoxifen complex in Proviron. Usually appointed by twenty to thirty milligrams of tamoxifen and no more than fifty milligrams Proviron. Joint reception of these drugs provides a remarkable effect.

 

This combination of drugs bodybuilders can greatly improve your results. Tamoxifen works well during a diet since it helps keeping the fat burning process. Lacking a direct property burn fat, the drug due to its exposure to antiestrogen helps to maintain a reduced level of fat in the body.

 

Tamoxifen should be taken in conjunction with the androgenic steroids or with different variations of testosterone. Athletes who have a tendency to increased accumulation in the body of water, or with a tendency to problems with mammary gland must be used this drug for any steroid treatment for prevention.

 

Since tamoxifen gives excellent results can take many bodybuilders androgenic steroids up until the start of the competition of the day, in combination with a diuretic. This course will give them the opportunity to appear on stage dried and elastic. Those athletes who have fat levels are already low, using tamoxifen get a great chance to significantly increase the density of the muscles.

 

Tamoxifen contributes to the number of units of high density cholesterol (HVP), capable of reducing the risk of atherosclerosis, therefore, it reduces greatly the risk of occurrence of cardiovascular diseases. This feature is very useful for athletes who are often faced with the disease. Another positive aspect is the fact that tamoxifen, a drug being soft, it manifests in the liver greater estrogenic activity. This feature has a positive effect on liver functions and the functioning of the whole organism.

 

However, along with all the advantages, tamoxifen numerous inherent disadvantages, which must be aware of every athlete, without exception, who wants to use this drug.

 

Tamoxifen bodybuilding – how to take on the FCT after a course?

Tamoxifen is a competitive inhibitor of peripheral estrogen receptor. And if earlier it was believed that the drug does not have the influence of estrogen, but today this view is totally rejected. In fact, the ratio of agonist and antagonist activity equal to 45/55. Tamoxifen is a chemically derived form triphenylethylene. The drug belongs to the group of sex hormones. Initially it was used for the treatment of cancer in women (breast cancer). But, undoubtedly, today Tamoxifen is much more common in sports and bodybuilding in particular.

 

It is no secret that the majority of steroids are exposed flavoring that is converted in to the female sex hormones – estrogens. This can lead to a variety of side effects, which is able to warn svoevremennyypriem Tamoxifen. Unlike other means such exposure, the substance is neither androgen or anabiotic.

 

Action Tamoxifen

 

  • The increase in power performance.
  • Increased hardness and muscle relief.
  • The increase in muscle mass. Tamoxifen is very popular in bodybuilding Argued that without it can not do any one victory in major competitions.
  • The marked anti-estrogen effects. The effect, which made so popular Tamoxifen. The higher dosage of AAC, the greater the need to compensate for estrogenic activity. Tamoxifen or analogues thereof at FCT after heavy courses practically mandatory.
  • The fight against fat.
  • Prevention of feminization.
  • Reducing the risk of developing atherosclerosis, the prevention of cardiovascular disease.
  • Improving liver.

Tamoxifen antiestrogen effects caused by blocking estrogen receptors (rather than the termination of the conversion of testosterone into estrogen, as many think). Preparation only freezes estrogenic activity, and does not prevent it entirely.

 

How to take Tamoxifen after the course

 

How to take Tamoxifen TamoksifenPriem after a course of steroids should be combined with an aromatase inhibitor, the most popular of which is Proviron (it is often used for the reason that it does not inhibit the production of growth hormone and inhibits aromatase, thereby increasing the concentration of anabolic hormones in the blood). Tamoxifen as a primary means of PCT is used in doses of 10 to 20 milligrams daily from the last week of the course and ending the second week of its completion. If Proviron is not accepted, Tamoxifen is included later – at 2 weeks, and ends 2-3 weeks after its cancellation. Read more

 

Please note that the highest levels of estrogen in the body occurs at the end of the first week of the course AAS. As for how to take Tamoxifen bodybuilding on a course of steroids, flavoring has no effect, it is recommended to add it only at the end of the cycle.

 

Side effects

 

The most common side effects of Tamoxifen associated with its pronounced antiestrogenic properties. Exceeding the recommended dose and / or duration of the course can cause female hair loss or total hair loss, flushing intense heat, itching, perineal pain in the bones; men – fever, dizziness, nausea. Because of the delay zhidkostimozhet disrupt the normal functioning of the kidneys. Also, sometimes there are bouts of depression, depression and drowsiness. Excessive intake is fraught with fatigue, constipation, and anorexia. You may experience inflammation of the retina, cataract, partial or complete loss of vision. Tamoxifen is sometimes accompanied by a rash on the skin. Cases of headache, changes in the cornea, unclear consciousness. Liver occur only in case of serious diseases of the body (such as hepatitis).

 

Reviews of Tamoxifen

 

Reviews TamoksifenOchen often expressed about the preparation of the athletes not as Tamoxifen for many years been used in post-menopausal women with estrogen-receptor-positive, and breast cancer patients. As for athletes, they are a marked anti-estrogen effects. Despite the wide range of possible side effects of Tamoxifen reviews indicate that adverse reactions are extremely rare. More info

 

Women athletes talk about the impossibility of use of the drug during pregnancy. In addition, it can prevent the implantation of the egg in the uterine wall. Reviews of tamoxifen on entry-level athletes are rare because amateurs are often bypassed by simple solo AAS courses that do not require FCT.

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Tamoxifen bodybuilding – application rates and side effects

Tamoxifen has the ability to deal with the excesses of estradiol, which occurs in the body due to the use of flavoring agents during hormone therapy and after its completion. After completing the course AAS’s own production of testosterone decreases significantly, and the body begins to produce instead of testosterone, estradiol, which finally destroys testosterone. But there are ways to combat these phenomena.

Buy tamoxifen

Tamoxifen, as well as Clomid may join estradiol receptors and block them. They block estrogen receptors, but have no effect on the levels of estrogen and the reduction is important not only to suppress the activity of estradiol and lower estrogen levels in the blood. This can be done with the help of anti-estrogen drugs such as Proviron.

Tamoxifen powerful Clomid several times. Therefore, the dosage of tamoxifen – 20-40 mg and Clomid – 50-100 mg. Research Clomid and tamoxifen have shown that is possible to increase the level of testosterone by 42% in 10 days if used tamoxifen 20 mg daily. A Clomid for this would take 150 mg per day.

Tamoxifen

Tenstosteron in the body is produced by exposure to the testes of luteinizing hormone (LH). The PH is, the more testosterone. LH produced by the pituitary gland and its production affects the hypothalamic gonadotropin-releasing hormone (GnRH). The hypothalamus regulates the production of GnRH depending on the level of testosterone and estradiol in the blood. In the production of GnRH it has a negative impact both too low and too high a level of estradiol. read more

Clomid increases LH only in the specified period of 10 minutes, and then it lowers it. Therefore, to use Clomid for more than 10 days is meaningless. Tamoxifen increases the PH 6 consecutive weeks.

In the blood estradiol and testosterone are often in the form of a bound. They are related to a particular protein – SHBG. This means that the bound form of any one of these hormones do not exert their activity. Clomid increases the level of SHBG in the blood, and tamoxifen – no. This is on one hand useful because estradiol is in a bound state, and therefore it is inactive, and on the other hand, also inactive and testosterone, which are already harmful.

The benefits of tamoxifen include the fact that this drug increases the level of high-density cholesterol. The second advantage stems from the fact that tamoxifen – a very mild estrogen, which significantly shows its estrogenic activity in the liver, and this has a positive effect on the entire body.

Clomid We still have one advantage over tamoxifen. Tamoxifen, although only slightly, but still reduce the possibility of developing a body of insulin-like growth factor (IGF-1), and Clomid, which manifests itself as estrogen in the liver are not so active, it has the disadvantage of a lesser degree.

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